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兰索拉唑中间体的研究进展
引用本文:徐俊,杨根生. 兰索拉唑中间体的研究进展[J]. 浙江化工, 2010, 41(6): 7-9
作者姓名:徐俊  杨根生
作者单位:浙江工业大学,药学院,浙江,杭州,310014
摘    要:介绍了抗胃溃疡新药兰索拉唑的重要中间体2-氯甲基-3-甲基-4-(2,2,2-三氟乙氧基)吡啶的各种合成方法,并评价了其优缺点,明确指出了一种最佳的合成方法。

关 键 词:兰索拉唑  中间体  合成  方法

Progress on Research of Lansoprazole Intermediates
XU Jun,YAN Gen-sheng. Progress on Research of Lansoprazole Intermediates[J]. Zhejiang Chemical Industry, 2010, 41(6): 7-9
Authors:XU Jun  YAN Gen-sheng
Affiliation:XU Jun, YAN Gen-sheng (College of Pharmaceutical Science,Zhejiang University of Technology,Hangzhou 310014,China)
Abstract:Synthesis methods for new drug intermediate of Lansoprazole peptic antiulcer were reviewed. Their advantages and disadvantages were evaluated. An optimum synthesis method was explicitly pointed out.
Keywords:ALansoprazole  intermediate  synthesis  method
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