| S-四嗪衍生物的合成及其生物活性初报 |
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| 引用本文： | 江银枝,陈洁,胡惟孝. S-四嗪衍生物的合成及其生物活性初报[J]. 现代农药, 2004, 3(3): 20-22 |
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| 作者姓名： | 江银枝 陈洁 胡惟孝 |
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| 作者单位： | 1. 浙江工业大学药学院,杭州,310014
2. 浙江省化工研究院南方农药创制中心,杭州,310000 |
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| 基金项目： | 国家自然科学基金(20272053)，浙江省自然科学基金资助(200016) |
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| 摘 要： | 利用2种路线合成了11种s-四嗪衍生物,并用熔点测定、IR、MS、1H NMR进行了确认,对未知化合物还进行了元素分析。对其中部分化合物进行了生物活性实验,发现有些化合物显示了较好的活性,同时发现烷基取代基的引入可以提高除草活性。
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| 关 键 词： | s-四嗪 衍生物 合成 分析 活性 除草 |
| 修稿时间： | 2003-11-27 |
Syntheses and Biological Activities of S-tetrazines |
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| Jiang Yinzhi Chen Jie Hu Weixiao. Syntheses and Biological Activities of S-tetrazines[J]. Modern Agrochemicals, 2004, 3(3): 20-22 |
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| Authors: | Jiang Yinzhi Chen Jie Hu Weixiao |
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| Affiliation: | Jiang Yinzhi1 Chen Jie2 Hu Weixiao1 |
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| Abstract: | Eleven derivatives of s-tetrazines were synthesized and characterized by m.p., IR , MS, 1H NMR and the elemental analysis. Seven among these compounds had been synthesized from hydrazine and nitrile in alcohol under refluxing by using S as catalysis. Four else had been synthesized from hydrazine and aldehyde without any catalysis. Some experiments were did on herbicide activity, and had found that activities of some compounds was good,especially 3,6-bis-benzyl-s-tetrazine. |
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| Keywords: | s-tetrazine derivative synthesize analysis activity herbicide |
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